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1.Discovery of N-(4-(Benzyloxy)-phenyl)-sulfonamide Derivatives as Novel Antagonists of the Human Androgen Receptor Targeting the Activation Function 2
Chai, Xin, Sun, Huiy
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Chai, Xin, Sun, Huiyong, Zhou, Wenfang, Chen, Changwei, Shan, Luhu, Yang, Yuhui, He, Junzhao, Pang, Jinping, Yang, Liu, Wang, Xinyue, Cui, Sunliang, Fu, Yaqin, Xu, Xiaohong, Xu, Lei, Yao, Xiaojun, Li, Dan, Hou, Tingjun
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Journal of Medicinal Chemistry[0022-2623],
Published 2022,
Volume 65,
Issue 3,
Pages 2507-2521
收錄情况:
WOS
SCOPUS
WOS核心合集引用: 6
2022影響因子:
7.3
发表年影響因子:
7.3
2.RELATION: A Deep Generative Model for Structure-Based De Novo Drug Design
Wang, MY, Hsieh, CY,
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Wang, MY, Hsieh, CY, Wang, JK, Wang, D, Weng, GQ, Shen, C, Yao, XJ, Bing, ZT, Li, HL, Cao, DS, Hou, TJ
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JOURNAL OF MEDICINAL CHEMISTRY[0022-2623],
Published 2022,
收錄情况:
WOS
SCOPUS
WOS核心合集引用: 18
2022影響因子:
7.3
发表年影響因子:
7.3
3.ChemistGA: A Chemical Synthesizable Accessible Molecular Generation Algorithm for Real-World Drug Discovery
Wang, JK, Wang, XR,
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Wang, JK, Wang, XR, Sun, HY, Wang, MY, Zeng, YD, Jiang, DJ, Wu, ZX, Liu, ZY, Liao, B, Yao, XJ, Hsieh, CY, Cao, DS, Chen, X, Hou, TJ
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JOURNAL OF MEDICINAL CHEMISTRY[0022-2623],
Published 2022,
Volume 65,
Issue 18,
Pages 12482-12496
收錄情况:
WOS
WOS核心合集引用: 3
2022影響因子:
7.3
发表年影響因子:
7.3
4.Structural Modification of Aminophenylarsenoxides Generates Candidates for Leukemia Treatment via Thioredoxin Reductase Inhibition
Song, ZL, Zhang, JM,
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Song, ZL, Zhang, JM, Xu, QH, Shi, DF, Yao, XJ, Fang, JG
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JOURNAL OF MEDICINAL CHEMISTRY[0022-2623],
Published 2021,
Volume 64,
Issue 21,
Pages 16132-16146
收錄情况:
WOS
SCOPUS
WOS核心合集引用: 15
2022影響因子:
7.3
发表年影響因子:
8.039